ʻO Reserpine kahi alkaloid indole i hoʻohana ʻia i ka mālama ʻana i ka hypertension a me ka psychosis. Ua unuhi mua ia mai ka mea kanu Serpentine. I kēia mau lā, no ka nui o nā hopena ʻaoʻao a me nā lāʻau lapaʻau hou ʻoi aku ka maikaʻi ma ka mākeke, ʻaʻole ʻo reserpine ke koho mua no ka mālama ʻana. Catecholamines (monoamine neurotransmitters) pāʻani koʻikoʻi i ka hoʻoponopono ʻana i ka puʻuwai puʻuwai, myocardial contractile ikaika a me peripheral resistance, a hoʻohana ka reserpine i kona hopena antihypertensive ma o ka ʻai ʻana i nā catecholamines mai nā hopena nerve sympathetic peripheral.
Hiki ke hoʻoheheʻe ʻia i loko o ka chloroform, dichloromethane, glacial acetic acid, hiki ke hoʻoheheʻe i loko o ka benzene, ethyl acetate, hiki ke hoʻoheheʻe ʻia i ka acetone, methanol, ethanol, ether, acetic acid a me citric acid solutions. Huli melemele ka hopena o ka reserpine ma hope o kekahi manawa, a he nui ka fluorescence, a hoʻonui ʻia ka fluorescence ma hope o ka hoʻohui ʻana a me ka hoʻolaha. ʻO ka Reserpine kahi kumu nāwaliwali. Hiki i ka Reserpine ke hoʻohaʻahaʻa i ke koko a me ka lohi o ka naʻau. He lohi, mālie a lōʻihi kāna hana. Loaʻa iā ia kahi hopena hoʻomaha lōʻihi ma ke kikowaena o ke kikowaena a he mea hoʻomaha maikaʻi.
Hoʻopilikia nui ka Reserpine i ka lawe ʻana o ka norepinephrine i loko o nā vesicle i nā hopena aʻalolo aloha, e hoʻohaʻahaʻa ʻia ai e ka monoamine oxidase a hoʻopau i ka mālama ʻana o nā norepinephrine, no laila e hoʻopilikia ai i ka lawe ʻana i nā neʻe aʻalolo sympathetic. ʻO kēia ka hopena i ka dilation vascular, hoʻemi i ke koko, a hoʻemi i ka puʻuwai puʻuwai. ʻO ka hoʻomaha ʻana a me ka hoʻopaʻa ʻana i ke kikowaena o ka ʻōnaehana ma muli paha o ke komo ʻana o reserpine i ka lolo a hoʻopau i ka waihona catecholamine waena. Hōʻike ka hopena hypotensive i loko o 1 mau hola ma hope o ka hoʻokele intravenous. Hoʻomaka ka hopena antihypertensive o ka mālama waha ma kahi o 1 pule ma hope o ka lawelawe ʻana a hiki i kona hopena kiʻekiʻe ma hope o 2-3 mau pule. Hoʻomau ka hopena no 3-4 mau pule ma hope o ka pau ʻana o ka mālama ʻana.
Loaʻa iā mākou nā hale hana kiʻekiʻe me ka pilina hohonu, hiki iā ia ke hāʻawi iā ʻoe i nā huahana kiʻekiʻe a me nā kumukūʻai hoʻokūkū. A hiki iā mākou ke hāʻawi i nā uku no nā kūʻai nui. A ke hui pū nei mākou me nā ʻoihana lawe ukana ʻoihana he nui, hiki ke hāʻawi i nā huahana me ka palekana a me ka maʻalahi i kou mau lima. ʻO ka manawa hoʻouna ma kahi o 3-20 mau lā ma hope o ka hōʻoia ʻana o ka uku.
Pilikino lāʻau
Hiki i nā anesthetics maʻamau ke hoʻonui i ka hopena antihypertensive o ka reserpine. I ka hui pū ʻana me ka ethanol a i ʻole nā mea hoʻopaneʻe o ka ʻōnaehana kikowaena, hiki ke hoʻonui ʻia ka hopena o ke kikowaena.
1. hui pū ʻia me nā lāʻau antihypertensive ʻē aʻe a i ʻole diuretics hiki ke hoʻoikaika i ka hopena antihypertensive, pono e hoʻoponopono ʻia ka nui; I ka hui pū me ka β-blocker, hiki ke hoʻonui i ka hopena hope;
2. hui pū ʻia me ka digitalis a i ʻole quinidine, hiki i nā kumu nui ke hoʻoulu i ka arrhythmia;
3. hui pū ʻia me ka levodopa hiki ke hoʻopau i ka dopamine, e alakaʻi ana i ka maʻi o Parkinson;
4. hui pū ʻia me nā lāʻau adrenergic indirect e like me ka ephedrine, amphetamine, a me nā mea ʻē aʻe, hiki ke hana i ka depletion mālama catecholamine, ke kāohi i ka hopena o nā lāʻau adrenergic;
5. hui pū me nā lāʻau adrenergic pololei e like me epinephrine, isoproterenol, norepinephrine, mehydroxyamine, deoxyadrenalin, etc., hiki ke hoʻolōʻihi i kona hopena;
6. hui pū me nā antidepressants tricyclic, ua nāwaliwali nā hopena o ka reserpine a me nā antidepressants;
7. hiki i ka barbiturates ke hoʻoikaika i ka hopena sedative waena o ka reserpine.
ʻO ka nui o ka lāʻau
ʻAʻohe lāʻau lapaʻau kūikawā ʻo Reserpine, ʻaʻole hiki ke hoʻopau ʻia e ka dialysis, ʻo nā ʻano lapaʻau he symptomatic a me ke kākoʻo ʻana. ʻO ka overdose ke kumu o ka hanu hanu, coma, ke koko haʻahaʻa, convulsions, a me ka hypothermia. I kēia manawa, pono e lawe ʻia ka hoʻomaʻemaʻe ʻōpū e hoʻoulu i ka luaʻi, ʻoiai ma hope o kekahi mau hola o ka lāʻau lapaʻau. Hoʻonoho ʻia nā maʻi me ka hypotension koʻikoʻi ma ke kūlana moe, ua hoʻokiʻekiʻe ʻia ko lākou mau wāwae, a ua mālama pono ʻia nā lāʻau epinephrine pololei e hoʻoikaika i ke koko. Hāʻawi ʻia ka inhalation oxygen a me ka hanu ʻana i nā poʻe maʻi me ke kaumaha hanu. Hoʻomaʻamaʻa nā lāʻau anticholinergic i nā hōʻailona ʻōpū; A hoʻoponopono i ka dehydration, electrolyte imbalance, hepatic coma, a me ka hypotension. Pono e nānā ʻia nā mea maʻi no ka liʻiliʻi o 72 mau hola no ka mea lōʻihi ka hana o ka reserpine. ʻO ke koko i ka pae ʻoluʻolu.
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