Sitagliptin is an oral antihyperglycemic of the dipeptidyl peptidase-4 inhibitor class. This enzyme-inhibiting drug is used either alone or in combination with other oral antihyperglycemic agents for treatment of diabetes mellitus type 2.The benefit of this medicine is its fewer side effects in the control of blood glucose values. While safety is its advantage, efficacy is often challenged as it is often recommended to be combined with other agents such as metformin.
Sitagliptin is a dipeptidyl peptidase-4 (DPP-4) inhibitor that controls blood glucose levels by protecting and enhancing endogenous enteroglycin.Glucose-dependent insulin-releasing peptides (GIP) and glucagon-like peptide-1 (GLP-1) are enteroglycins released in response to dietary intake.
GLP-1 and GIP can increase insulin synthesis and release from islet β cells through intracellular signaling pathways. GLP-1 can also reduce glucagon secretion from islet α cells and reduce hepatic glucose production.However, both GLP-1 and GIP are rapidly metabolized by DPP-4, resulting in the loss of their insulin-promoting effect.
Vi har mange højkvalitetsfabrikker med dybt samarbejde, som kan give dig produkter af høj kvalitet og konkurrencedygtige priser. Og vi kan også give rabat ved bulkkøb. Og vi samarbejder med mange professionelle speditionsfirmaer, kan levere produkter sikkert og problemfrit til dine hænder. Leveringstiden er omkring 3-20 dage efter bekræftelse af betaling.
Vare | Test Standard | Testing Result | |
CBD | Not less than (NLT) 99.5% 99.9% | ||
THC | Not detected | Undetected | |
Assay | Method HPLC calculated on the anhydrous basis limit of quotation (LOQ) 0.8ppm | ||
Udseende | Hvidt pulver | White powder | |
Identifikation | In the recorded chromatograms under the determination of the substance, retention time of the main peak of the solution should be consistent with the retention of time of the main peak of the reference solution | Overholder | |
Smeltepunkt | 65~66ºC | 65.5ºC | |
Tab ved tørring | NMT 1.0% | 0.21% | |
Residual solvents | Ethanol NMT 400ppm Heptane NMT 400ppm |
1.92ppm 256.0ppm |
|
Heavy Mental | NMT 20ppm | Overholder | |
Microbial Limite Test | Method: Plate Counting | ||
Total aerobic bacteria count | NMT 1000cfu/g | Overholder | |
Combined molds and yeast | NMT 100cfu/g | Overholder | |
E. Coli | Not detacted per gram | Overholder | |
Salmanella | Not detacted per 10 gram | Overholder | |
Conclusion: Conform the testing result is qualified |
1. Er du en fabrik eller en handelsvirksomhed?
Vi er en virksomhed, der integrerer industri og handel, og leverer one-stop service.OEM kunne accepteres.
2. Giver du prøver? Er det gratis eller ekstra?
Gratis prøver. Prøvens fragtgebyr skal betales ved din side.
3. Har du nogen certifikater relateret til kvalitetskontrol?
ISO 9001:2008 certificering for at sikre kvalitet.
4. Hvad skal jeg give for at få et tilbud?
Pls informer os om den produkttype, du har brug for, ordremængde, adresse og specifikke krav. Tilbuddet vil blive lavet til din reference i tide.
5. Hvilken slags betalingsmetode foretrækker du? Hvilken slags vilkår accepteres?
Accepterede leveringsbetingelser: FOB, CFR, CIF, EXW;
Accepted Payment Currency:USD;EUR
Accepteret betalingstype: T/T, Western Union; Paypal, Trade Assurance.
Talt sprog: engelsk.
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