LGD-4033 is a non-steroidal oral, selective androgen receptor modulator in healthy young adults
LGD-4033 is a non-steroidal oral, selective androgen receptor modulator in healthy young people
Sinemizi-mveliso emininzi ekumgangatho ophezulu enentsebenziswano enzulu, enokubonelela ngeemveliso ezikumgangatho ophezulu kunye namaxabiso akhuphisanayo. Kwaye sinako ukunika izaphulelo zokuthengwa kwezinto ezininzi.Kwaye siyasebenzisana neenkampani ezininzi zokuthunyelwa kwempahla, zinokuzisa iimveliso ngokukhuselekileyo nangokutyibilikayo ezandleni zakho. Ixesha lokuhambisa limalunga neentsuku ezi-3-20 emva kokuqinisekiswa kwentlawulo.
Molecular Formula | C14H12F6N2O |
Molar Mass | 338.25 |
Density | 1.45±0.1 g/cm3(Predicted) |
Indawo yokunyibilika | 108 - 111°C |
Boling Point | 439.9±45.0 °C(Predicted) |
Solubility | Acetone (Slightly), Chloroform (Slightly, Heated), Methanol (Slightly) |
Imbonakalo | A crystalline solid |
Color | White to Pale Beige |
pKa | 12.06±0.20(Predicted) |
Storage Condition | Hygroscopic, -20°C Freezer, Under inert atmosphere |
Uzinzo | Hygroscopic |
In vivo study | In animal models, LGD-4033 has anabolic activity in muscle, suppressive resorption and anabolic activity in bone, and is more selective in muscle than in prostate. At the concentrations tested, LGD-4033 was safe and well-tolerated, with a long elimination half-life of about 24-36 hours and a linear pharmacokinetics profile. |
1. Ngaba uyifektri okanye inkampani yokurhweba?
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Iisampuli zasimahla. Umrhumo womthwalo wesampulu kufuneka uhlawulwe ecaleni kwakho.
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ISO 9001:2008 isiqinisekiso sokuqinisekisa umgangatho.
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