LGD-4033 is a non-steroidal oral, selective androgen receptor modulator in healthy young adults
LGD-4033 is a non-steroidal oral, selective androgen receptor modulator in healthy young people
Loaʻa iā mākou nā hale hana kiʻekiʻe me ka pilina hohonu, hiki iā ia ke hāʻawi iā ʻoe i nā huahana kiʻekiʻe a me nā kumukūʻai hoʻokūkū. A hiki iā mākou ke hāʻawi i nā uku no nā kūʻai nui. A ke hui pū nei mākou me nā ʻoihana lawe ukana ʻoihana he nui, hiki ke hāʻawi i nā huahana me ka palekana a me ka maʻalahi i kou mau lima. ʻO ka manawa hoʻouna ma kahi o 3-20 mau lā ma hope o ka hōʻoia ʻana o ka uku.
Molecular Formula | C14H12F6N2O |
Molar Mass | 338.25 |
Density | 1.45±0.1 g/cm3(Predicted) |
Lae hehee | 108 - 111°C |
Boling Point | 439.9±45.0 °C(Predicted) |
Solubility | Acetone (Slightly), Chloroform (Slightly, Heated), Methanol (Slightly) |
Ka nana aku | A crystalline solid |
Color | White to Pale Beige |
pKa | 12.06±0.20(Predicted) |
Storage Condition | Hygroscopic, -20°C Freezer, Under inert atmosphere |
Paʻa | Hygroscopic |
In vivo study | In animal models, LGD-4033 has anabolic activity in muscle, suppressive resorption and anabolic activity in bone, and is more selective in muscle than in prostate. At the concentrations tested, LGD-4033 was safe and well-tolerated, with a long elimination half-life of about 24-36 hours and a linear pharmacokinetics profile. |
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