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LGD-4033 CAS 1165910-22-4

LGD-4033 CAS 1165910-22-4

 

  • Izina RY'IGICURUZWA:

    LGD-4033 CAS 1165910-22-4

  • Icyiciro:

    Urwego rwa farumasi

  • Ibyiza:

    ifu yera

  • Gupakira:

    25kg / ingoma

  • MOQ:

    1 kilo

  • Ububiko:Ahantu humye
  • Ubuzima bwa Shelf:Imyaka 2


Ibisobanuro

Etiquetas

Ibisobanuro ku bicuruzwa

LGD-4033 is a non-steroidal oral, selective androgen receptor modulator in healthy young adults

Gusaba

LGD-4033 is a non-steroidal oral, selective androgen receptor modulator in healthy young people

Ibyiza

Dufite inganda nyinshi zo mu rwego rwo hejuru hamwe nubufatanye bwimbitse, zishobora kuguha ibicuruzwa byiza kandi nibiciro byapiganwa. Turashobora kandi gutanga kugabanyirizwa kugura byinshi.Kandi turafatanya namasosiyete menshi yohereza ibicuruzwa byumwuga, birashobora gutanga ibicuruzwa neza kandi neza mumaboko yawe. Igihe cyo gutanga ni iminsi 3-20 nyuma yo kwemeza ko wishyuye.

 

Ibisobanuro
Molecular Formula C14H12F6N2O
Molar Mass 338.25
Density 1.45±0.1 g/cm3(Predicted)
Ingingo yo gushonga 108 - 111°C
Boling Point 439.9±45.0 °C(Predicted)
Solubility Acetone (Slightly), Chloroform (Slightly, Heated), Methanol (Slightly)
Kugaragara A crystalline solid
Color White to Pale Beige
pKa 12.06±0.20(Predicted)
Storage Condition Hygroscopic, -20°C Freezer, Under inert atmosphere
Igihagararo Hygroscopic
In vivo study In animal models, LGD-4033 has anabolic activity in muscle, suppressive resorption and anabolic activity in bone, and is more selective in muscle than in prostate. At the concentrations tested, LGD-4033 was safe and well-tolerated, with a long elimination half-life of about 24-36 hours and a linear pharmacokinetics profile.

 

Kohereza no kwishyura

 

Ibibazo

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