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Tesofensine

Good quality Tesofensine CAS 195875-84-4

 

  • Product name:

    Tesofensine

  • Giredhi:

    Pharmaceutical/Cosmetic grade

  • Properties:

    white powder

  • Packing:

    25kg / chigubhu

  • MOQ:

    1 kilo

  • Kuchengeta:Nzvimbo Yakaoma yakaoma
  • Sherufu hupenyu:2 years


Details

Tags

Product Description

Tesofensine (NS-2330) is a triple monoamine reuptake inhibitor inducing a potent inhibition of the re-uptake process in the synaptic cleft of the neurotransmitters dopamine (DA; IC50=6.5 nM), norepinephrine (NE;IC50=1.7 nM), and serotonin (5-HT;IC50=11 nM), and with potentials as an anti-obesity agent[1]. Tesofensine is a CNS acting anti-obesity agent[2].

Application

Tesofensine (NS-2330) is a triple monoamine reuptake inhibitor inducing a potent inhibition of the re-uptake process in the synaptic cleft of the neurotransmitters dopamine (DA; IC50=6.5 nM), norepinephrine (NE;IC50=1.7 nM), and serotonin (5-HT;IC50=11 nM), and with potentials as an anti-obesity agent. Tesofensine is a CNS acting anti-obesity agent.

Zvakanakira

Tine mafekitori akawanda emhando yepamusoro nekubatana kwakadzama, ayo anogona kukupa zvigadzirwa zvemhando yepamusoro nemitengo yemakwikwi. Uye isu tinogonawo kupa zvidzikiso pakutenga kwakawanda. Uye isu tinobatirana nemakambani mazhinji ehunyanzvi ekutakura zvinhu, anogona kuendesa zvigadzirwa zvakachengeteka uye zvakanaka kumaoko ako. Nguva yekutumira inenge 3-20 mazuva mushure mekusimbiswa kwekubhadhara.

 

Tsanangudzo
Product Name: tesofensine
Synonyms: (1S,3S,4R,5R)-3-(3,4-dichlorophenyl)-4-(ethoxymethyl)-8-methyl-8-azabicyclo[3.2.1]octane;(1R,2R,3S,5S)-3-(3,4-Dichlorophenyl)-2-(ethoxymethyl)-8-methyl-8-azabicyclo[3.2.1]octane;Tesofensine-13C-d3;8-Azabicyclo[3.2.1]octane, 3-(3,4-dichlorophenyl)-2-(ethoxymethyl)-8-methyl-, (1R,2R,3S,5S)-
CAS: 195875-84-4
MF: C17H23Cl2NO
MW: 328.28
EINECS:  
Product Categories:  
Mol File: 195875-84-4.mol
tesofensine Structure
 
tesofensine Chemical Properties
Boiling point  396.6±42.0 °C(Predicted)
density  1.161±0.06 g/cm3(Predicted)
kuchengetedza temp.  Store at -20°C
solubility  DMF: 2 mg/mL,DMSO: 1 mg/mL,Ethanol: Slightly soluble,PBS (pH 7.2): 0.14 mg/mL
form  A solid
pka 10.46±0.60(Predicted)
color  White to off-white

 

Kutumira uye kubhadhara


 

FAQ

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2. Unopa mienzaniso here? Ndeyemahara here kana kuti yakawedzerwa?
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3. Iwe une chero zvitupa zvine chekuita nekutonga kwemhando?
ISO 9001:2008 certification kuti ive nechokwadi chemhando.

4. Chii chandinofanira kupa kuti ndiwane quotation?
Pls inotizivisa nezverudzi rwechigadzirwa chaunoda, huwandu hwekuraira, kero uye zvakananga zvinodiwa.The quotation ichaitwa kuti utarise nguva yako.

5. Ndeipi nzira yekubhadhara yaunoda? Ndeapi mazwi anogamuchirwa?
Mitemo Yekutumira Inogamuchirwa: FOB, CFR, CIF, EXW;
Mari Yekubhadhara Yakagamuchirwa: USD;
Rudzi rwekubhadhara rwakagamuchirwa: T / T, Western Union; Paypal, Trade Assurance.
Mutauro Unotaurwa:Chirungu.

 

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