Tesofensine (NS-2330) is a triple monoamine reuptake inhibitor inducing a potent inhibition of the re-uptake process in the synaptic cleft of the neurotransmitters dopamine (DA; IC50=6.5 nM), norepinephrine (NE;IC50=1.7 nM), and serotonin (5-HT;IC50=11 nM), and with potentials as an anti-obesity agent[1]. Tesofensine is a CNS acting anti-obesity agent[2].
Tesofensine (NS-2330) is a triple monoamine reuptake inhibitor inducing a potent inhibition of the re-uptake process in the synaptic cleft of the neurotransmitters dopamine (DA; IC50=6.5 nM), norepinephrine (NE;IC50=1.7 nM), and serotonin (5-HT;IC50=11 nM), and with potentials as an anti-obesity agent. Tesofensine is a CNS acting anti-obesity agent.
Manana orinasa avo lenta maro miaraka amin'ny fiaraha-miasa lalina, izay afaka manome anao vokatra avo lenta sy ny vidiny mifaninana. Ary afaka manome fihenam-bidy ho an'ny fividianana betsaka ihany koa izahay.Ary miara-miasa amin'ny orinasa mpitatitra entana matihanina maro izahay, afaka manatitra vokatra soa aman-tsara sy milamina amin'ny tananao. Delivery fotoana dia tokony ho 3-20 andro aorian'ny fanamafisana ny fandoavam-bola.
Product Name: | tesofensine |
Synonyms: | (1S,3S,4R,5R)-3-(3,4-dichlorophenyl)-4-(ethoxymethyl)-8-methyl-8-azabicyclo[3.2.1]octane;(1R,2R,3S,5S)-3-(3,4-Dichlorophenyl)-2-(ethoxymethyl)-8-methyl-8-azabicyclo[3.2.1]octane;Tesofensine-13C-d3;8-Azabicyclo[3.2.1]octane, 3-(3,4-dichlorophenyl)-2-(ethoxymethyl)-8-methyl-, (1R,2R,3S,5S)- |
CAS: | 195875-84-4 |
MF: | C17H23Cl2NO |
MW: | 328.28 |
EINECS: | |
Product Categories: | |
Mol File: | 195875-84-4.mol |
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tesofensine Chemical Properties |
Teboka mangotraka | 396.6±42.0 °C(Predicted) |
hakitroky | 1.161±0.06 g/cm3(Predicted) |
temp. | Store at -20°C |
solubility | DMF: 2 mg/mL,DMSO: 1 mg/mL,Ethanol: Slightly soluble,PBS (pH 7.2): 0.14 mg/mL |
-KARAZANY | A solid |
pka | 10.46±0.60(Predicted) |
loko | White to off-white |
1. Orinasa ve ianao sa orinasa mpivarotra?
Izahay dia compnay mampiditra ny indostria sy ny varotra, manome serivisy tokana. Azo ekena ny OEM.
2. Manome santionany ve ianao? Maimaimpoana ve sa fanampiny?
Santionany maimaim-poana.Ny sandan'ny entana santionany dia mila aloa eo anilanao.
3. Manana taratasy fanamarinana mifandraika amin'ny fanaraha-maso kalitao ve ianao?
ISO 9001: 2008 fanamarinana mba hiantohana ny kalitao.
4. Inona no tokony homeko mba hahazoana teny nindramina?
Pls ampahafantaro anay ny karazana vokatra ilainao, ny habetsaky ny baiko, ny adiresy ary ny fepetra takiana manokana.
5. Inona no fomba fandoavam-bola tianao? Karazana fepetra inona no ekena?
Fepetra fanaterana ekena: FOB, CFR, CIF, EXW;
Vola fandoavana ekena:USD;
Karazana fandoavam-bola ekena: T / T, Western Union; Paypal, Trade Assurance.
Fiteny ampiasaina: Anglisy.
Ny sokajy vokatra